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N-(4-Fluorobenzyl)-3-hydroxy-9,9-dimethyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrazino[1,2-a]pyrimidine-2-carboxamides a novel class of potent HIV-1 integrase inhibitors.

Petrocchi A, Jones P, Rowley M, Fiore F, Summa V. (2009)
Bioorg Med Chem Lett. 2009 Aug 1;19(15):4245-9.

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